product summary
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company name :
Tocris Bioscience
product type :
chemical
product name :
VTP 27999 trifluoroacetate
catalog :
5563
quantity :
10 mg
price :
172 USD
more info or order :
Tocris Bioscience product webpage
product information
brand :
Tocris
master code :
5563
SKU :
5563/10
product name :
VTP 27999 trifluoroacetate
description :
Highly potent and selective renin inhibitor
target :
Additional Synthetic Protease Inhibitors
category :
Small Molecules
unit size :
10 mg
purity :
97%
observed molecular weight :
639.1
url print :
?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
Highly potent and selective renin inhibitor (IC50 = 0.47 nM). Displays 1000-fold selectivity over related and unrelated off-targets. Blocks renin-stimulated ERK1/2 phosphorylation in vascular smooth muscle cells. Exhibits a different mode of action to aliskiren (Cat. No. 5491).
catalog number base :
5563
product keywords :
VTP 27999 trifluoroacetate highly potent selective renin inhibitors inhibits Other Proteases 5563,
extended description :
Highly potent and selective renin inhibitor
chemical name text :
Methyl N-[2-[(R)-(3-Chlorophenyl)[(3R)-1-[[[(2S)-2-(methylamino)-3-[(3R)-tetrahydro-2H-pyran-3-yl]propyl]amino]carbonyl]-3-piperidinyl]methoxy]ethyl]carbamate trifluoroacetate
formula :
C 26 H 41 ClN 4 O 5 .CF 3 CO 2 H
formula text :
C26H41ClN4O5.CF3CO2H
cas num :
1013937-63-7
2020 USD :
172
2021 USD :
172 USD
storage :
Store at -20°C
more info or order :
Tocris Bioscience product webpage
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK