5563/10 | Tocris Bioscience 5563/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5563/10

catalog :

5563/10

quantity :

10 mg

price :

193 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5563 - VTP 27999 trifluoroacetate C26H41ClN4O5.CF3CO2H CAS No. 1013937-63-7

product information

master code :

5563

SKU :

5563/10

product name :

VTP 27999 trifluoroacetate

unit size :

10 mg

description :

Highly potent and selective renin inhibitor

target :

Additional Synthetic Protease Inhibitors

category :

Small Molecules

purity :

97%

observed molecular weight :

639.1

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VTP 27999 trifluoroacetate is a highly potent and selective renin inhibitor (IC50 = 0.47 nM). Displays 1000-fold selectivity over related and unrelated off-targets. Blocks renin-stimulated ERK1/2 phosphorylation in vascular smooth muscle cells. Exhibits a different mode of action to aliskiren (Cat. No. 5491).

top caption :

Highly potent and selective renin inhibitor

extended description :

Highly potent and selective renin inhibitor

chemical name text :

Methyl N-[2-[(R)-(3-Chlorophenyl)[(3R)-1-[[[(2S)-2-(methylamino)-3-[(3R)-tetrahydro-2H-pyran-3-yl]propyl]amino]carbonyl]-3-piperidinyl]methoxy]ethyl]carbamate trifluoroacetate

formula :

C26H41ClN4O5.CF3CO2H

formula text :

C26H41ClN4O5.CF3CO2H

cas num :

1013937-63-7

USD :

193 USD

product details :

Highly potent and selective renin inhibitor

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage