Perlapine | Tocris Bioscience 5549 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Perlapine

catalog :

5549

quantity :

10 mg (also 50 mg)

price :

147 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Weston M, Kaserer T, Wu A, Mouravlev A, Carpenter J, Snowball A, et al. Olanzapine: A potent agonist at the hM4D(Gi) DREADD amenable to clinical translation of chemogenetics. Sci Adv. 2019;5:eaaw1567 pubmed publisher

product information

brand :

Tocris

master code :

5549

SKU :

5549/10

product name :

Perlapine

description :

Potent hM3Dq and hM4Di DREADD agonist in vitro

target :

DREADD Activators

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

291.39

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent muscarinic DREADD agonist (pEC50 values are 8.38, 8.08 and 7.27 for hM1Dq, hM3Dq and hM4Di in vitro , respectively). Exhibits 10,000-fold selectivity for hM3Dq over hM3 receptors.

catalog number base :

5549

product keywords :

Perlapine potent selective hM3Dq DREADD agonists antagonism designer receptors drugs muscarinic receptors activators chemogenetics DREADDs Non-selective Muscarinics 5549, Chemogenetics

extended description :

Potent hM3Dq and hM4Di DREADD agonist in vitro

chemical name text :

6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

formula :

C 19 H 21 N 3

formula text :

C19H21N3

cas num :

11/3/77

2020 USD :

144

2021 USD :

147 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage