5549/10 | Tocris Bioscience 5549/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5549/10

catalog :

5549/10

quantity :

10 mg (also 50 mg)

price :

185 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Weston M, Kaserer T, Wu A, Mouravlev A, Carpenter J, Snowball A, et al. Olanzapine: A potent agonist at the hM4D(Gi) DREADD amenable to clinical translation of chemogenetics. Sci Adv. 2019;5:eaaw1567 pubmed publisher

image

image 1 :

Cat.No. 5549 - Perlapine C19H21N3 CAS No. 1977-11-3

product information

master code :

5549

SKU :

5549/10

product name :

Perlapine

unit size :

10 mg (also 50 mg)

description :

Potent hM3Dq and hM4Di DREADD agonist in vitro

target :

DREADD Activators

category :

Small Molecules

purity :

99%

observed molecular weight :

291.39

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Perlapine is a potent muscarinic DREADD agonist (pEC50 values are 8.38, 8.08 and 7.27 for hM1Dq, hM3Dq and hM4Di in vitro , respectively). Exhibits 10,000-fold selectivity for hM3Dq over hM3 receptors.

top caption :

Potent hM3Dq and hM4Di DREADD agonist in vitro

extended description :

Potent hM3Dq and hM4Di DREADD agonist in vitro

chemical name text :

6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

formula :

C19H21N3

formula text :

C19H21N3

cas num :

11/3/77

USD :

185 USD

product details :

Potent hM3Dq and hM4Di DREADD agonist in vitro

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage