5546/10 | Tocris Bioscience 5546/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5546/10

catalog :

5546/10

quantity :

10 mg (also 50 mg)

price :

167 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5546 - NI 57 C19H17N3O4S

product information

master code :

5546

SKU :

5546/10

product name :

NI 57

unit size :

10 mg (also 50 mg)

description :

Potent and selective BRPF bromodomain inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

383.42

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

NI 57 is a potent and selective BRPF bromodomain inhibitor (Kd values are 31, 108 and 408 nM, for BRPF1B, 2 and 3, respectively, which exhibits >32-fold selectivity for BRPFs over BRD9 and other non-Class IV bromodomains. NI 57 inhibits RANKL-induced differentiation of primary murine bone marrow cells and human primary monocytes into osteoclasts.

top caption :

Potent and selective BRPF bromodomain inhibitor

extended description :

Potent and selective BRPF bromodomain inhibitor

chemical name text :

4-Cyano-N-(1,3-dimethyl-2-oxo-1,2-dihydroquinolin-6-yl)-2-methoxybenzene-1-sulfonamide

formula :

C19H17N3O4S

formula text :

C19H17N3O4S

cas num :

1883548-89-7

USD :

167 USD

product details :

Potent and selective BRPF bromodomain inhibitor

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage