LP 99 | Tocris Bioscience 5496 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LP 99

catalog :

5496

quantity :

25 mg

price :

1039 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5496

SKU :

5496/25

product name :

LP 99

description :

Selective BRD7 and BRD9 inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

unit size :

25 mg

purity :

98%

observed molecular weight :

516.05

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective BRD7 and BRD9 inhibitor (Kd values are 99 and 909 nM, respectively). Exhibits selectivity for BRD7/9 over a panel of 48 bromodomains (at 10 M). Inhibits interactions with histones H3.3 and H4 at low micromolar concentrations. Decreases the level of IL-6 secreted from LPS-stimulated THP-1 cells. Negative control ent-LP 99 (Cat.No. 5497) also available.

catalog number base :

5496

product keywords :

LP99 selective BRD7 BRD9 bromodomain inhibitors inhibits Bromodomains 5496,

extended description :

Selective BRD7 and BRD9 inhibitor

chemical name text :

N-[(2R,3S)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide

formula :

C 26 H 30 ClN 3 O 4 S

formula text :

C26H30ClN3O4S

cas num :

1808951-93-0

2020 USD :

999

2021 USD :

1039 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage