5496/5 | Tocris Bioscience 5496/5 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5496/5

catalog :

5496/5

quantity :

5 mg (also 25 mg)

price :

285 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5496 - LP 99 C26H30ClN3O4S CAS No. 1808951-93-0

product information

master code :

5496

SKU :

5496/5

product name :

LP 99

unit size :

5 mg (also 25 mg)

description :

Selective BRD7 and BRD9 inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

516.05

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

LP 99 is a selective BRD7 and BRD9 inhibitor (Kd values are 99 and 909 nM, respectively) that exhibits selectivity for BRD7/9 over a panel of 48 bromodomains (at 10 M). LP 99 inhibits interactions with histones H3.3 and H4 at low micromolar concentrations, and decreases the level of IL-6 secreted from LPS-stimulated THP-1 cells, in vitro . A negative control for LP 99, ent-LP 99 (Cat.No. 5497), is also available.

top caption :

Selective BRD7 and BRD9 inhibitor

extended description :

Selective BRD7 and BRD9 inhibitor

chemical name text :

N-[(2R,3S)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide

formula :

C26H30ClN3O4S

formula text :

C26H30ClN3O4S

cas num :

1808951-93-0

USD :

285 USD

product details :

Selective BRD7 and BRD9 inhibitor

storage :

Store at -20░C

more info or order :

Tocris Bioscience product webpage