product summary
Loading...
company name :
Tocris Bioscience
product type :
chemical
product name :
AC 4
catalog :
5464
quantity :
10 mg (also 50 mg)
price :
211 USD
more info or order :
product information
brand :
Tocris
master code :
5464
SKU :
5464/10
product name :
AC 4
description :
Photoswitchable TRPV1 channel blocker
target :
TRPV Antagonists
category :
Small Molecules
unit size :
10 mg (also 50 mg)
purity :
98%
observed molecular weight :
514.56
url print :
?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
Photoswitchable TRPV1 channel blocker (IC50 = 3.1 M). Acts as an antagonist in trans conformation during voltage gated activation. Also acts as an antagonist in the cis formation during capsaicin-induced TRPV1 currents. Switches conformation from cis to trans at 440 nm and trans to cis at 360 nm. Allows photoswitchable antagonist and an agonist to be applied at the same time.
catalog number base :
5464
product keywords :
Photoswitchable TRPV1 channel blockers transient receptor potential vanilloids ligands Photoswitchable Ligands TRPV 5464,
extended description :
Photoswitchable TRPV1 channel blocker
chemical name text :
1,3,4,5-Tetrahydro-7,8-dihydro-N-[2-[4-[2-[4-(trifluoromethyl)phenyl]diazenyl]phenyl]ethyl]-2H-2-benzazepine-2-carbothioamide
formula :
C 26 H 25 F 3 N 4 O 2 S
formula text :
C26H25F3N4O2S
cas num :
1459809-09-6
2020 USD :
234
2021 USD :
211 USD
storage :
Store at -20°C
more info or order :
company information

Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com800-343-7475
headquarters: UK
browse more products
questions and comments