VU 0469650 hydrochloride | Tocris Bioscience 5379 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

VU 0469650 hydrochloride

catalog :

5379

quantity :

10 mg (also 50 mg)

price :

208 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5379

SKU :

5379/10

product name :

VU 0469650 hydrochloride

description :

Potent and selective negative allosteric modulator of mGlu1 receptors

target :

Group I mGluR Modulators

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

400.94

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective negative allosteric modulator of mGlu1 (IC50 = 99 nM). Exhibits 100-fold selectivity for mGlu1 over mGlu2-8 and 68 other GPCRs, ion channels, kinases and transporters. Brain penetrant.

catalog number base :

5379

product keywords :

VU0469650 hydrochloride modulators metabotropic glutamate receptor mGlu1 mGluR1 allosteric negative potent selective NAMs Glutamate (Metabotropic) Group I Receptors 5379,

extended description :

Potent and selective negative allosteric modulator of mGlu1 receptors

chemical name text :

3-[(3R)-3-Methyl-4-(tricyclo[3.3.1.13,7]dec-1-ylcarbonyl)-1-piperazinyl]-2-pyridinecarbonitrile hydrochloride

formula :

C 22 H 28 N 4 O.HCl

formula text :

C22H28N4O.HCl

cas num :

1443748-47-7

2020 USD :

201

2021 USD :

208 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage