5379/10 | Tocris Bioscience 5379/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5379/10

catalog :

5379/10

quantity :

10 mg (also 50 mg)

price :

233 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5379 - VU 0469650 hydrochloride C22H28N4O.HCl CAS No. 1443748-47-7

product information

master code :

5379

SKU :

5379/10

product name :

VU 0469650 hydrochloride

unit size :

10 mg (also 50 mg)

description :

Potent and selective negative allosteric modulator of mGlu1 receptors

target :

Group I mGluR Modulators

category :

Small Molecules

purity :

98%

observed molecular weight :

400.94

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

VU 0469650 hydrochloride is a potent and selective negative allosteric modulator of mGlu1 (IC50 = 99 nM). Exhibits 100-fold selectivity for mGlu1 over mGlu2-8 and 68 other GPCRs, ion channels, kinases and transporters. Brain penetrant.

top caption :

Potent and selective negative allosteric modulator of mGlu1 receptors

extended description :

Potent and selective negative allosteric modulator of mGlu1 receptors

chemical name text :

3-[(3R)-3-Methyl-4-(tricyclo[3.3.1.13,7]dec-1-ylcarbonyl)-1-piperazinyl]-2-pyridinecarbonitrile hydrochloride

formula :

C22H28N4O.HCl

formula text :

C22H28N4O.HCl

cas num :

1443748-47-7

USD :

233 USD

product details :

Potent and selective negative allosteric modulator of mGlu1 receptors

storage :

Store at +4░C

more info or order :

Tocris Bioscience product webpage