5367/10 | Tocris Bioscience 5367/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

5367/10

catalog :

5367/10

quantity :

10 mg (also 50 mg)

price :

191 USD

more info or order :

Tocris Bioscience product webpage

image

image 1 :

Cat.No. 5367 - SGC 707 C16H18N4O2

product information

master code :

5367

SKU :

5367/10

product name :

SGC 707

unit size :

10 mg (also 50 mg)

description :

Potent and selective allosteric inhibitor of PRMT3

target :

Protein Arginine Methyltransferase Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

298.34

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SGC 707 is a potent allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3) (IC50 = 31 nM). Inhibits PRMT3-mediated methyltransferase activity in vitro . Displays 100-fold selectivity against 31 other methyltransferases and 250 other non-epigenetic targets. Decreases H4R3me2a levels in HEK293 cells in vitro . . Negative control also available.

top caption :

Potent and selective allosteric inhibitor of PRMT3

extended description :

Potent and selective allosteric inhibitor of PRMT3

chemical name text :

1-(Isoquinolin-6-yl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl] urea

formula :

C16H18N4O2

formula text :

C16H18N4O2

cas num :

1687736-54-4

USD :

191 USD

product details :

Potent and selective allosteric inhibitor of PRMT3

storage :

Store at +4░C

more info or order :

Tocris Bioscience product webpage