BMS 564929 | Tocris Bioscience 5274/5 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BMS 564929

catalog :

5274/5

quantity :

5 mg

price :

159 USD

citations: 1

Reference
Schlezinger J, Heiger Bernays W, Webster T. Predicting the Activation of the Androgen Receptor by Mixtures of Ligands Using Generalized Concentration Addition. Toxicol Sci. 2020;177:466-475 pubmed publisher

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

5274

SKU :

5274/5

product name :

BMS 564929

description :

Highly potent and muscle-selective androgen receptor (AR) agonist

target :

Androgen Receptor Agonists

unit size :

5 mg

category :

Small Molecules

purity :

98%

storage :

Store at -20°C

observed molecular weight :

305.72

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BMS 564929 is a highly potent and selective androgen receptor (AR) agonist (EC50 = 0.44 nM). Exhibits selectivity for ARs over estrogen, glucocorticoid and mineralocorticoid receptors and no significant binding to steroid hormone binding globulin or aromatase. Also exhibits selectivity for muscle over prostate ARs. Active in vivo and orally bioavailable.

product keywords :

BMS564929 highly potent muscle-selective androgen receptor AR agonist orally bioavailable Androgen Receptor 5274,

extended description :

Highly potent and muscle-selective androgen receptor (AR) agonist

chemical name text :

2-Chloro-3-methyl-4-[(7R,7aS)-tetrahydro-7-hydroxy-1,3-dioxo-1H-pyrrolo[1,2-c]imidazol-2(3H)-yl]benzonitrile

formula :

C14H12ClN3O3

formula text :

C14H12ClN3O3

cas num :

627530-84-1

USD :

157

USD 2025 :

159 USD

product details :

Highly potent and muscle-selective androgen receptor (AR) agonist