GSK 137647 | Tocris Bioscience 5257 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GSK 137647

catalog :

5257

quantity :

10 mg (also 50 mg)

price :

113 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5257

SKU :

5257/10

product name :

GSK 137647

description :

Potent and selective FFA4 (GPR120) agonist

target :

Free Fatty Acid Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

305.39

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective FFA4 (GPR120) agonist (pEC50 values are 6.3, 6.2 and 6.1 at the human, mouse and rat receptor, respectively). Exhibits 100-fold selectivity against a panel of 61 targets including FFA1, FFA2 and FFA3. Enhances glucose-stimulated insulin secretion in MIN6 cells. Induces intracellular calcium accumulation in U2OS cells; this activity is inhibited by AH 7614 (Cat. No. 5256).

catalog number base :

5257

product keywords :

GSK137647 Free fatty acid receptor 4 diabetes potent and selective FFA4 GPR120 agonist Free Fatty Acid Receptors 5257,

extended description :

Potent and selective FFA4 (GPR120) agonist

chemical name text :

4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide

formula :

C 16 H 19 NO 3 S

formula text :

C16H19NO3S

cas num :

349085-82-1

2020 USD :

109

2021 USD :

113 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage