AH 7614 | Tocris Bioscience 5256 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AH 7614

catalog :

5256

quantity :

10 mg (also 50 mg)

price :

115 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Kishikawa A, Kitaura H, Kimura K, Ogawa S, Qi J, Shen W, et al. Docosahexaenoic Acid Inhibits Inflammation-Induced Osteoclast Formation and Bone Resorption in vivo Through GPR120 by Inhibiting TNF-α Production in Macrophages and Directly Inhibiting Osteoclast Formation. Front Endocrinol (Lausanne). 2019;10:157 pubmed publisher
Chen Y, Lin Y, Sun C, Huang T, Yip H, Chen Y. Extracorporeal shockwave against inflammation mediated by GPR120 receptor in cyclophosphamide-induced rat cystitis model. Mol Med. 2018;24:60 pubmed publisher

product information

brand :

Tocris

master code :

5256

SKU :

5256/10

product name :

AH 7614

description :

Selective FFA4 (GPR120) antagonist

target :

Free Fatty Acid Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

351.42

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective free fatty acid receptor 4 (FFA4/GPR120) antagonist (pIC50 values are 7.1 and 4.6 for human FFA4 and FFA1 receptors respectively). Inhibits linoleic acid and GSK 137647A -induced intracellular calcium accumulation in U2OS osteosarcoma cells expressing the FFA4 receptor.

catalog number base :

5256

product keywords :

AH7614 selective free fatty acid 4 FFA4 receptor antagonist GPR120 Free Fatty Acid Receptors 5256,

extended description :

Selective FFA4 (GPR120) antagonist

chemical name text :

4-Methyl-N-9H-xanthen-9-yl-benzenesulfonamide

formula :

C 20 H 17 NO 3 S

formula text :

C20H17NO3S

cas num :

6/3/26

2020 USD :

110

2021 USD :

115 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage