chemical

CC4

5236

10 mg (also 50 mg)

147 USD

5236

5236/10

CC4

High affinity and subtype-selective 6 2 and 4 2 nAChR partial agonist

Additional Nicotinic (a4b2) Receptor Compounds

Small Molecules

10 mg (also 50 mg)

98%

406.52

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

High affinity and subtype selective 6 2 and 4 2 partial agonist (Ki values are 12 and 26nM for rat 6 2 and 4 2 receptors respectively). Has low affinity for 3 4 and 7 receptors (Ki values are 4.8 and 13 M for human 3 4 and rat 7 receptors respectively). Stimulates dopamine release from striatal slices in vitro . Attenuates nicotine-induced self-administration and conditional place preference in rats.

5236

CC4 high affinity subtype selective partial agonist acetylcholine nicotinic receptors alpha4beta2 a4b2 4 2 alpha6beta3 a6b3 6 3 Nicotinic (a4b2) Receptors Nicotinic Receptors (Other Subtypes) 5236,

High affinity and subtype-selective 6 2 and 4 2 nAChR partial agonist

(1R,5S)-1,2,3,4,5,6-Hexahydro-3-[2-[(1R,5S)-1,5,6,8-tetrahydro-8-oxo-1,5-methano-2H-pyrido[1,2-a][1,5]diazocin-3(4H)-yl]ethyl]-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one

C 24 H 30 N 4 O 2

C24H30N4O2

492-02-4

144

147 USD

Store at +4°C