This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.
product summary
company name :
Tocris Bioscience
product type :
chemical
product name :
NIBR 189
catalog :
5203/10
quantity :
10 mg (also 50 mg)
price :
243 USD
product information
brand :
Tocris
master code :
5203
SKU :
5203/10
product name :
NIBR 189
unit size :
10 mg (also 50 mg)
seo description :
Potent and selective EBI2 (GPR183) receptor antagonist
target :
Orphan 7-TM Receptor Antagonists
category :
Small Molecules
purity :
99%
observed molecular weight :
429.31
url print :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
details of functionality :
NIBR 189 is a potent and selective EBI2 (GPR183) receptor antagonist (IC50 values are 11 and 15 nM for human and mouse EBI2 receptors respectively). Exhibits selectivity for EBI2 over a panel of other receptors, enzymes and transporters. Blocks oxysterol-induced migration of U937 monocyte cells. Orally bioavailable.
top caption :
Potent and selective EBI2 (GPR183) receptor antagonist
extended description :
Potent and selective EBI2 (GPR183) receptor antagonist
chemical name text :
(2E)-3-(4-Bromophenyl)-1-[4-4-methoxybenzoyl)-1-piperazinyl]-2-propene-1-one
formula :
C21H21BrN2O3
formula text :
C21H21BrN2O3
cas num :
1599432-08-2
USD :
243 USD
product details :
Potent and selective EBI2 (GPR183) receptor antagonist
storage :
Store at +4░C
company information
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
headquarters: UK