ASP 7663 | Tocris Bioscience 5178/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

ASP 7663

catalog :

5178/10

quantity :

10 mg (also 50 mg)

price :

246 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Blaha I, López Oliva M, Martínez M, Recio P, Agis Torres A, Martinez A, et al. Bladder Dysfunction in an Obese Zucker Rat: The Role of TRPA1 Channels, Oxidative Stress, and Hydrogen Sulfide. Oxid Med Cell Longev. 2019;2019:5641645 pubmed publisher
Ko M, Ganzen L, Coşkun E, Mukadam A, Leung Y, van Rijn R. A critical evaluation of TRPA1-mediated locomotor behavior in zebrafish as a screening tool for novel anti-nociceptive drug discovery. Sci Rep. 2019;9:2430 pubmed publisher

image

image 1 :

Cat.No. 5178 - ASP 7663 C14H14FNO3 CAS No. 1190217-35-6

product information

brand :

Tocris

master code :

5178

SKU :

5178/10

rank :

0.061

product name :

ASP 7663

description :

Selective TRPA1 activator

target :

TRPA1 Activators

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

ASP 7663 is a selective TRPA1 activator (EC50 values are ~0.5 M in human, mouse and rat). Displays little or no affinity at more than 60 other related receptors, channels and enzymes. Stimulates 5-HT release from QGP-1 cells. Exhibits an abdominal analgesic effect in vivo . Orally bioavailable.

extended description :

Selective TRPA1 activator

chemical name text :

(2E)-2-[7-Fluoro-1,2-dihydro-1-(2-methylpropyl)-2-oxo-3H-indol-3-ylidene]acetic acid

formula :

C 14 H 14 FNO 3

formula text :

C14H14FNO3

cas num :

1190217-35-6

USD :

246 USD

product details :

Selective TRPA1 activator

storage :

Store the unopened product at 2 - 8 °C. Do not use past expiration date.

more info or order :

Tocris Bioscience product webpage