TG 4-155 | Tocris Bioscience 5052 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

TG 4-155

catalog :

5052

quantity :

10 mg (also 50 mg)

price :

221 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Cuesto G, Jordán Álvarez S, Enriquez Barreto L, Ferrús A, Morales M, Acebes A. GSK3β inhibition promotes synaptogenesis in Drosophila and mammalian neurons. PLoS ONE. 2015;10:e0118475 pubmed publisher

product information

brand :

Tocris

master code :

5052

SKU :

5052/10

product name :

TG 4-155

description :

High affinity and selective EP2 receptor antagonist

target :

Prostanoid Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

394.46

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity and selective EP2 receptor antagonist (KB values are 2.4 and 34.5 nM for EP2 and DP1 receptors respectively). Exhibits 500-fold selectivity for EP2 over other prostanoid receptors. Inhibits butaprost-induced proinflammatory cytokine production, cell proliferation and invasion of PC-3 cells in vitro .

catalog number base :

5052

product keywords :

TG4-155 high affinity selective EP2 prostanoid receptors antagonists Prostanoid Receptors 5052,

extended description :

High affinity and selective EP2 receptor antagonist

chemical name text :

(2E)-N-[2-(2-Methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide

formula :

C 23 H 26 N 2 O 4

formula text :

C23H26N2O4

cas num :

1164462-05-8

2020 USD :

216

2021 USD :

221 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage