TC-E 5001 | Tocris Bioscience 5049 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

TC-E 5001

catalog :

5049

quantity :

10 mg (also 50 mg)

price :

149 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

5049

SKU :

5049/10

product name :

TC-E 5001

description :

Potent tankyrase inhibitor

target :

Tankyrase Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

409.46

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Dual tankyrase (TNKS) inhibitor (Kd values are 79 and 28 nM for TNKS1 and TNKS2 respectively, IC50 = 33 nM for TNKS2) that is devoid of activity at PARP1 and PARP2 (IC50 19 M). Inhibits Wnt signaling and stabilizes Axin2 levels.

catalog number base :

5049

product keywords :

TC-E5001 TNKS1 TNKS2 tankyrase inhibitors inhibits wnt signaling signalling Poly(ADP-ribose) Polymerase Tankyrase 5049,

extended description :

Potent tankyrase inhibitor

chemical name text :

3-(4-Methoxyphenyl)-5-[[[4-(4-methoxyphenyl)-5-methyl-4H-1,2,4-triazol-3-yl]thio]methyl]-1,2,4-oxadiazole

formula :

C 20 H 19 N 5 O 3 S

formula text :

C20H19N5O3S

cas num :

865565-29-3

2020 USD :

149

2021 USD :

149 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage