PEAQX tetrasodium salt | Tocris Bioscience 5018/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PEAQX tetrasodium salt

catalog :

5018/10

quantity :

10 mg

price :

336 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Malci A, Lin X, Sandoval R, Gundelfinger E, Naumann M, Seidenbecher C, et al. Ca2+ signaling in postsynaptic neurons: Neuroplastin-65 regulates the interplay between plasma membrane Ca2+ ATPases and ionotropic glutamate receptors. Cell Calcium. 2022;106:102623 pubmed publisher
Mares P, Tsenov G, Kubova H. Anticonvulsant Action of GluN2A-Preferring Antagonist PEAQX in Developing Rats. Pharmaceutics. 2021;13: pubmed publisher

image

image 1 :

Cat.No. 5018 - PEAQX tetrasodium salt C17H13BrN3Na4O5P

product information

brand :

Tocris, a Bio-Techne brand

catalog number base :

5018

SKU :

5018/10

product name :

PEAQX tetrasodium salt

description :

Potent and GluN2A-selective NMDA antagonist

target :

NMDA Receptor Antagonists

unit size :

10 mg

category :

Small Molecules

purity :

98%

storage :

Store at -20°C

observed molecular weight :

542.14

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

PEAQX tetrasodium salt is a potent NMDA receptor antagonist (IC50 = 8 nM). Exhibits 100-fold selectivity for hGluN2A (formally hNR2A) containing receptors over hGluN2B (hNR2B). Anticonvulsant in vivo . . Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions .

product keywords :

NVP-AAM 077 anticonvulsants potent selective NMDA subtype antagonists antagonism 459836-30-7 2102348-87-6 NMDA Receptors 5018,

extended description :

Potent and GluN2A-selective NMDA antagonist

chemical name text :

[[[(1S)-1-(4-Bromophenyl)ethyl]amino](1,2,3,4-tetrahydro-2,3-dioxo-5-quinoxalinyl)methyl] phosphonic acid tetrasodium salt

formula :

C17H13BrN3Na4O5P

formula text :

C17H13BrN3Na4O5P

USD :

332

USD 2025 :

336 USD

product details :

Potent and GluN2A-selective NMDA antagonist

more info or order :

Tocris Bioscience product webpage