Eplivanserin hemifumarate | Tocris Bioscience 4958/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Eplivanserin hemifumarate

catalog :

4958/10

quantity :

10 mg (also 50 mg)

price :

205 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

4958

SKU :

4958/10

product name :

Eplivanserin hemifumarate

Description :

Potent and selective 5-HT2A antagonist

target :

5-HT2A Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

386.42

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Eplivanserin hemifumarate is a potent and selective 5-HT2A antagonist (IC50 values are 5.8 and 120 and >100 nM for 5-HT2A, 5-HT2B and 5-HT2C, respectively). Attenuates cocaine-induced hyperactivity. Increases dopamine (DA) release in rat medial prefrontal cortex (mPFC); potentiates haloperidol-induced DA release in the mPFC and nucleus accumbens.

extended description :

Potent and selective 5-HT2A antagonist

chemical name text :

(1Z,2E)-1-(2-Fluorophenyl)-3-(4-hydroxyphenyl)-2-propen-1-one O-[2-(dimethylamino)ethyl]oxime hemifumarate

formula :

C 19 H 21 FN 2 O 2 .0.5C 4 H 4 O 4

formula text :

C19H21FN2O2.0.5C4H4O4

cas num :

130580-02-8

USD :

205 USD

product details :

Potent and selective 5-HT2A antagonist

alt names :

SR-46349 hemifumarate, SR-46349B

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage