OXF BD 02 | Tocris Bioscience 4928/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

OXF BD 02

catalog :

4928/10

quantity :

10 mg (also 50 mg)

price :

228 USD

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

4928

SKU :

4928/10

product name :

OXF BD 02

Description :

Selective BRD4(1) inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

295.33

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

OXF BD 02 is a selective inhibitor of the first bromodomain of BRD4 (BRD4(1)) (IC50 = 382 nM). Exhibits 2-3-fold selectivity for BRD4(1) over the CBP bromodomain and has little affinity for a range of other bromodomains. Reduces viability of lung adenocarcinoma cell lines and attenuates proliferation of MV-4-11 leukemia cells. Cell permeable.

extended description :

Selective BRD4(1) inhibitor

chemical name text :

3-(3,5-Dimethyl-4-isoxazolyl)-5-hydroxy- -phenylbenzenemethanol

formula :

C 18 H 17 NO 3

formula text :

C18H17NO3

cas num :

1429129-68-9

USD :

228 USD

product details :

Selective BRD4(1) inhibitor

storage :

Store at +4°C