I-CBP 112 | Tocris Bioscience 4891 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

I-CBP 112

catalog :

4891

quantity :

10 mg (also 50 mg)

price :

289 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

4891

SKU :

4891/10

product name :

I-CBP 112

description :

Selective CBP/p300 BRD inhibitor

target :

Bromodomain Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

468.59

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

CBP/p300 bromodomain inhibitor (IC50 values are 0.142-0.17 and 0.625 M for CBP and p300 respectively). Selective for CBP and p300 over ATAD2, BAZ2B, BRD2(2), BRD4(1), PB1(5), PCAF, PHIP(2) and TIF1 bromodomains in a BLI assay. Accelerates FRAP recovery in cells at a concentration of 1 M.

catalog number base :

4891

product keywords :

I-CBP112 CREBBP EP300 bromodomains selective inhibitors inhibits chemical probes SGC epigenetics structural genomics consortium Bromodomains Histone Acetyltransferases 4891,

extended description :

Selective CBP/p300 BRD inhibitor

chemical name text :

1-[7-(3,4-Dimethoxyphenyl)-9-[[(3S)-1-methylpiperidin-3-yl]methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one

formula :

C 27 H 36 N 2 O 5

formula text :

C27H36N2O5

cas num :

1640282-31-0

2020 USD :

280

2021 USD :

289 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage