H2L 5765834 | Tocris Bioscience 4870 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

H2L 5765834

catalog :

4870

quantity :

10 mg (also 50 mg)

price :

219 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Kittaka H, Uchida K, Fukuta N, Tominaga M. Lysophosphatidic acid-induced itch is mediated by signalling of LPA5 receptor, phospholipase D and TRPA1/TRPV1. J Physiol. 2017;595:2681-2698 pubmed publisher

product information

brand :

Tocris

master code :

4870

SKU :

4870/10

product name :

H2L 5765834

description :

LPA1,3,5 antagonist

target :

Lysophosphatidic Acid (LPA) Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

404.33

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Antagonist of the lysophosphatidic acid receptors LPA1, LPA5 and LPA3 (IC50 values are 94, 463 and 752 nM respectively). Exhibits no effect at LPA2 or LPA4 receptors.

catalog number base :

4870

product keywords :

H2L5765834 lysophosphatidic acid receptors LPA1 LPA3 LPA5 antagonists Lysophosphatidic Acid Receptors 4870,

extended description :

LPA1,3,5 antagonist

chemical name text :

2,3-Dihydro-2-[3-(4-nitrophenoxy)phenyl]-1,3-dioxo-1H-isoindole-5-carboxylic acid

formula :

C 21 H 12 N 2 O 7

formula text :

C21H12N2O7

cas num :

420841-84-5

2020 USD :

212

2021 USD :

219 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage