Gue 1654 | Tocris Bioscience 4742/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Gue 1654

catalog :

4742/10

quantity :

10 mg (also 50 mg)

price :

151 USD

citations: 1

Reference
Nogueras Ortiz C, Roman Vendrell C, Mateo Semidey G, Liao Y, Kendall D, Yudowski G. Retromer stops beta-arrestin 1-mediated signaling from internalized cannabinoid 2 receptors. Mol Biol Cell. 2017;28:3554-3561 pubmed publisher

product information

brand :

Tocris

master code :

4742

SKU :

4742/10

product name :

Gue 1654

target :

G Protein (Heterotrimeric) Inhibitors

category :

Small Molecules

unit sizes :

10 mg (also 50 mg)

purity :

97%

observed molecular weight :

447.6

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Gue 1654 is an oxoeicosanoid receptor 1 (OXE-R) modulator. Selectively inhibits G but not G i signaling upon activation of the G i- heterotrimer by OXE-R. Inhibits G -mediated opening of GIRK1/2 channels in HEK293 cells.

extended description :

Selective inhibitor of OXE-R G / signaling

chemical name text :

N-[7-(Methylthio)benzo[1,2-d:4,3-d ]bisthiazol-2-yl]- -phenylbenzeneacetamide

formula :

C 23 H 17 N 3 OS 3

formula text :

C23H17N3OS3

cas num :

397290-30-1

USD :

151 USD

product details :

Selective inhibitor of OXE-R G / signaling

storage :

Store at +4°C