SB 674042 | Tocris Bioscience 4673/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SB 674042

catalog :

4673/10

quantity :

10 mg (also 50 mg)

price :

377 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

4673

SKU :

4673/10

rank :

0.061

product name :

SB 674042

description :

Potent and selective non-peptide OX1 antagonist

target :

OX1 Receptor Antagonists

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SB 674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM). Exhibits 100-fold selectivity for OX1 over OX2 receptors. Has no effect at serotonergic, dopaminergic, adrenergic or purinergic receptors. Inhibits orexin 1-induced Ca2+ mobilization in CHO-DG44 cells stably transfected with the OX1 receptor.

extended description :

Potent and selective non-peptide OX1 antagonist

chemical name text :

[5-(2-Fluorophenyl)-2-methyl-4-thiazolyl][2(S)-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl-1-pyrrolidinyl]methanone

formula :

C 24 H 21 FN 4 O 2 S

cas num :

483313-22-0

USD :

377 USD

product details :

Potent and selective non-peptide OX1 antagonist

storage :

Store the unopened product at 2 - 8 °C. Do not use past expiration date.

more info or order :

Tocris Bioscience product webpage