PTAC oxalate | Tocris Bioscience 4533 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PTAC oxalate

catalog :

4533

quantity :

10 mg (also 50 mg)

price :

144 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Wang Y, Zuo Z, Zhang M, Feng Z, Yan M, Li X. The Analgesic Effects of (5R,6R)6-(3-Propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1] Octane on a Mouse Model of Neuropathic Pain. Anesth Analg. 2017;124:1330-1338 pubmed publisher

product information

brand :

Tocris

master code :

4533

SKU :

4533/10

product name :

PTAC oxalate

description :

Muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes

target :

Additional Non-selective Muscarinic Products

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

359.46

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Muscarinic receptor ligand. Displays partial agonist activity at M2 and M4 receptors; exhibits antagonist effects at M1, M3 and M5 receptors (Ki values are 2.8, 0.2, 0.6, 0.2 and 0.8 nM respectively). Displays selectivity for muscarinic receptors over a range of neurotransmitter receptors and ion channels. Inhibits firing rate of dopaminergic cells in the limbic ventral tegmental area after acute administration, without binding to dopamine receptors.

catalog number base :

4533

product keywords :

PTAC antipsychotics schizophrenia selective muscarinic partial agonists antagonists M1 M2 M3 M4 M5 Non-selective Muscarinics 4533,

extended description :

Muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes

chemical name text :

(1R,5R,6R)-6-[4-(Propylthio)-1,2,5-thiadiazol-3-yl]-1-azabicyclo[3.2.1]octane oxalate

formula :

C 12 H 19 N 3 S 2 .C 2 H 2 O 4

formula text :

C12H19N3S2.C2H2O4

cas num :

201939-40-4

2020 USD :

160

2021 USD :

144 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage