SHA 68 | Tocris Bioscience 4510 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

SHA 68

catalog :

4510

quantity :

10 mg (also 50 mg)

price :

223 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Ruzza C, Ferrari F, Guerrini R, Marzola E, Preti D, Reinscheid R, et al. Pharmacological profile of the neuropeptide S receptor: Dynamic mass redistribution studies. Pharmacol Res Perspect. 2018;6:e00445 pubmed publisher

product information

brand :

Tocris

master code :

4510

SKU :

4510/10

product name :

SHA 68

description :

Selective Neuropeptide S receptor antagonist

target :

Neuropeptide S Receptor Antagonist

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

445.49

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Selective neuropeptide S receptor (NPSR) antagonist (IC50 values are 22.0 and 23.8 nM for human NPSR Asn107 and Ile107 variants respectively). Displays no activity against a range of 14 GPCRs, including vasopressin and oxytocin receptors.

catalog number base :

4510

product keywords :

SHA68 neuropeptides S NPSRs NPS antagonists selective Neuropeptide S Receptors 4510, Neuropeptide-S Receptor, NPSR1

extended description :

Selective Neuropeptide S receptor antagonist

chemical name text :

N-[(4-Fluorophenyl)methyl]tetrahydro-3-oxo-1,1-diphenyl-3H-oxazolo[3,4-a]pyrazine-7(1H)-carboxamide

formula :

C 26 H 24 FN 3 O 3

formula text :

C26H24FN3O3

cas num :

847553-89-3

2020 USD :

214

2021 USD :

223 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage