4510/10 | Tocris Bioscience 4510/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

4510/10

catalog :

4510/10

quantity :

10 mg (also 50 mg)

price :

281 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Wang C, Xin L, Cai C, Cong C, Xie J, Kong X, et al. Neuropeptide S Displays as a Key Neuromodulator in Olfactory Spatial Memory. Chem Senses. 2020;45:195-202 pubmed publisher
Ruzza C, Ferrari F, Guerrini R, Marzola E, Preti D, Reinscheid R, et al. Pharmacological profile of the neuropeptide S receptor: Dynamic mass redistribution studies. Pharmacol Res Perspect. 2018;6:e00445 pubmed publisher

product information

master code :

4510

SKU :

4510/10

product name :

SHA 68

unit size :

10 mg (also 50 mg)

description :

Selective Neuropeptide S receptor antagonist

target :

Neuropeptide S Receptor Antagonists

category :

Small Molecules

purity :

98%

observed molecular weight :

445.49

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

SHA 68 is a selective neuropeptide S receptor (NPSR) antagonist (IC50 values are 22.0 and 23.8 nM for human NPSR Asn107 and Ile107 variants respectively). Displays no activity against a range of 14 GPCRs, including vasopressin and oxytocin receptors.

top caption :

Selective Neuropeptide S receptor antagonist

extended description :

Selective Neuropeptide S receptor antagonist

chemical name text :

N-[(4-Fluorophenyl)methyl]tetrahydro-3-oxo-1,1-diphenyl-3H-oxazolo[3,4-a]pyrazine-7(1H)-carboxamide

formula :

C26H24FN3O3

formula text :

C26H24FN3O3

cas num :

847553-89-3

USD :

281 USD

product details :

Selective Neuropeptide S receptor antagonist

storage :

Store at +4░C

more info or order :

Tocris Bioscience product webpage