Cercosporamide | Tocris Bioscience 4500/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

Cercosporamide

catalog :

4500/500

quantity :

500µg

price :

195 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

OC1=CC(O)=C(C(N)=O)C3=C1[C@@]2(C)C(O3)=CC(O)=C(C(C)=O)C2=O

Cat Number :

4500/500

Product Name :

Cercosporamide

Cas Number :

[131436-22-1]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

195 USD

Primary Category :

Enzymes

Secondary Category :

Kinases

Tertiary Category :

MAPK Family

Primary Action :

Potent Mnk2 inhibitor

Biological Description :

Potent inhibitor of MAP-kinase interacting kinase-2 (Mnk2) and JAK3 (IC50 values are 11, 31 and 116 nM for Mnk2, JAK3 and Mnk1 respectively). Blocks eIF4E phosphorylation; exhibits antiproliferative and proapoptotic activity in cancer cells in vitro. Also inhibits Pkc1. Orally bioavailable.

Formula :

C16H13NO7

Molwt :

331.28

more info or order :

Tocris Bioscience product webpage