GPBAR-A | Tocris Bioscience 4478 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

GPBAR-A

catalog :

4478

quantity :

10 mg (also 50 mg)

price :

220 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Kowal J, Haanes K, Christensen N, Novak I. Bile acid effects are mediated by ATP release and purinergic signalling in exocrine pancreatic cells. Cell Commun Signal. 2015;13:28 pubmed publisher

product information

brand :

Tocris

master code :

4478

SKU :

4478/10

product name :

GPBAR-A

description :

GPBA receptor (TGR5) agonist

target :

GPBA Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

484.37

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

GPBA receptor agonist. Upregulates GLP-1 secretion from intestinal cultures. Increases MQAE-fluorescence suggesting a decrease in intracellular chloride concentration in gallbladder epithelial cells.

catalog number base :

4478

product keywords :

TGR5 agonists g-protein bile acid receptors GPBA GPBAR GPBA Receptors 4478,

extended description :

GPBA receptor (TGR5) agonist

chemical name text :

4-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-6-(2-fluorophenyl)-4,5-dihydro-pyrido[3,2-f]-1,4-oxazepin-3(2H)-one

formula :

C 23 H 15 F 7 N 2 O 2

formula text :

C23H15F7N2O2

cas num :

877052-79-4

2020 USD :

244

2021 USD :

220 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage