PHP 501 trifluoroacetate | Tocris Bioscience 4466 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PHP 501 trifluoroacetate

catalog :

4466

quantity :

10 mg (also 50 mg)

price :

244 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
LeÃ³n S, Barroso A, VÃ¡zquez M, GarcÃa Galiano D, Manfredi Lozano M, Ruiz Pino F, et al. Direct Actions of Kisspeptins on GnRH Neurons Permit Attainment of Fertility but are Insufficient to Fully Preserve Gonadotropic Axis Activity. Sci Rep. 2016;6:19206 pubmed publisher

product information

brand :

Tocris

master code :

4466

SKU :

4466/10

product name :

PHP 501 trifluoroacetate

description :

Potent GABAA antagonist

target :

GABA-A Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

433.42

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent GABAA antagonist (Ki = 0.0028 M at rat GABAA receptors; IC50 = 0.024 M at human 1 2 2 GABAA-expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.

catalog number base :

4466

product keywords :

GABAA receptors antagonists potent PHP501 GABAA Receptors 4466,

extended description :

Potent GABAA antagonist

chemical name text :

4-(5-[1,1 -Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate

formula :

C 20 H 21 N 3O .CF 3 CO 2 H

formula text :

C20H21N3O.CF3CO2H

cas num :

1781880-44-1

2020 USD :

244

2021 USD :

244 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage