Bicifadine hydrochloride | Tocris Bioscience 4357/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Bicifadine hydrochloride

catalog :

4357/10

quantity :

10 mg (also 50 mg)

price :

144 USD

product information

brand :

Tocris

MasterCode :

4357

SKU :

4357/10

product name :

Bicifadine hydrochloride

unit sizes :

10 mg (also 50 mg)

description :

Noradrenalin, 5-HT and dopamine re-uptake inhibitor

target :

Adrenergic Transporter Inhibitors

category :

Small Molecules

purity :

98%

observed molecular weight :

209.72

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Bicifadine hydrochloride is a potent antagonist of the noradrenalin transporter (IC50 = 55 nM); also displays antagonist activity at the 5-HT and dopamine transporters (IC50 values are 117 nM and 910 nM respectively). Orally active. Exhibits antinociceptive and antiallodynic activity in rodent models of acute, persistent, and chronic pain.

extended description :

Noradrenalin, 5-HT and dopamine re-uptake inhibitor

chemical name text :

1-(4-Methylphenyl)-3-azabicyclo[3.1.0]hexane hydrochloride

formula :

C 12 H 15 N.HCl

formula text :

C12H15N.HCl

cas num :

66504-75-4

USD :

144 USD

product details :

Noradrenalin, 5-HT and dopamine re-uptake inhibitor

storage :

Desiccate at RT