AR-M 1000390 hydrochloride | Tocris Bioscience 4335/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

AR-M 1000390 hydrochloride

catalog :

4335/10

quantity :

10 mg (also 50 mg)

price :

240 USD

citations: 3

Reference
Radoux Mergault A, Oberhauser L, Aureli S, Gervasio F, Stoeber M. Subcellular location defines GPCR signal transduction. Sci Adv. 2023;9:eadf6059 pubmed publisher
Mann A, Liebetrau S, Klima M, Dasgupta P, Massotte D, Schulz S. Agonist-induced phosphorylation bar code and differential post-activation signaling of the delta opioid receptor revealed by phosphosite-specific antibodies. Sci Rep. 2020;10:8585 pubmed publisher
Stoeber M, Jullié D, Lobingier B, Laeremans T, Steyaert J, Schiller P, et al. A Genetically Encoded Biosensor Reveals Location Bias of Opioid Drug Action. Neuron. 2018;98:963-976.e5 pubmed publisher

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

4335

SKU :

4335/10

product name :

AR-M 1000390 hydrochloride

Description :

Low-internalizing agonist

target :

delta Opioid Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

97%

observed molecular weight :

384.94

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

AR-M 1000390 hydrochloride is a non-peptidic, low-internalizing -selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

extended description :

Low-internalizing agonist

chemical name text :

N,N-Diethyl-4-(phenyl-4-piperidinylidenemethyl)-benzamide hydrochloride

formula :

C 23 H 28 N 2 O.HCl

formula text :

C23H28N2O.HCl

cas num :

209808-47-9

USD :

240 USD

product details :

Low-internalizing agonist

storage :

Store at -20°C