PSB 0777 ammonium salt | Tocris Bioscience 4334/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PSB 0777 ammonium salt

catalog :

4334/10

quantity :

10 mg (also 50 mg)

price :

311 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Navarro G, Gonzalez A, Campanacci S, Rivas Santisteban R, Reyes Resina I, Casajuana Martin N, et al. Experimental and computational analysis of biased agonism on full-length and a C-terminally truncated adenosine A2A receptor. Comput Struct Biotechnol J. 2020;18:2723-2732 pubmed publisher
Wolska N, Kassassir H, Luzak B, Watala C, Rozalski M. Adenosine Receptor Agonists Increase the Inhibition of Platelet Function by P2Y12 Antagonists in a cAMP- and Calcium-Dependent Manner. Pharmaceuticals (Basel). 2020;13: pubmed publisher

product information

brand :

Tocris

catalog number base :

4334

SKU :

4334/10

product name :

PSB 0777 ammonium salt

units size :

10 mg (also 50 mg)

description :

Potent adenosine A2A agonist

target :

Adenosine A2a Receptor Agonists

category :

Small Molecules

purity :

97%

observed molecular weight :

500.55

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

PSB 0777 ammonium salt is a potent adenosine A2A receptor full agonist (Ki = 44.4 nM for rat brain striatal A2A receptors). Exhibits subtype selectivity for A2A receptors over A1, A2B and A3 receptors (Ki 10 000 nM for rat A1, human A2B and human A3 receptors). Potentiates acetylcholine-induced contractions in ex vivo rat ileum/jejunum segments.

top caption :

Potent adenosine A2A agonist

extended description :

Potent adenosine A2A agonist

chemical name text :

4-[2-[(6-Amino-9-b-D-ribofuranosyl-9H-purin-2-yl)thio]ethyl]benzenesulfonic acid ammonium salt

formula :

C18H20N5O7S2.NH4

formula text :

C18H20N5O7S2.NH4

cas num :

2122196-16-9

USD :

311 USD

product details :

Potent adenosine A2A agonist

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage