Gisadenafil besylate | Tocris Bioscience 4165/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Gisadenafil besylate

catalog :

4165/10

quantity :

10 mg (also 50 mg)

price :

204 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Silva J, Polesskaya O, Knight W, Zheng J, Granger M, Lopez T, et al. Transient hypercapnia reveals an underlying cerebrovascular pathology in a murine model for HIV-1 associated neuroinflammation: role of NO-cGMP signaling and normalization by inhibition of cyclic nucleotide phosphodiesterase-5. J Neuroinflammation. 2012;9:253 pubmed publisher

product information

brand :

Tocris

master code :

4165

SKU :

4165/10

rank :

0.061

product name :

Gisadenafil besylate

description :

Potent PDE5 inhibitor; orally bioavailable

target :

Phosphodiesterase Inhibitors

category :

Small Molecules

sizes available :

10 mg (also 50 mg)

url print :

?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Gisadenafil besylate is a potent PDE5 inhibitor (IC50 = 1.23 nM). Shows 100-fold selectivity for PDE5 over PDE6. Orally bioavailable.

extended description :

Potent PDE5 inhibitor; orally bioavailable

chemical name text :

5-[2-Ethoxy-5-[(4-ethyl-1-piperazinyl)sulfonyl]-3-pyridinyl]-3-ethyl-2,6-dihydro-2-(2-methoxyethyl)-7H-pyrazolo[4,3-d]pyrimidin-7-one benzenesulfonate

formula :

C 23 H 33 N 7 O 5 S.C 6 H 6 O 3 S

formula text :

C23H33N7O5S.C6H6O3S

cas num :

334827-98-4

USD :

204 USD

product details :

Potent PDE5 inhibitor; orally bioavailable

alt names :

UK 369003

storage :

Store the unopened product at room temperature. Do not use past expiration date.

more info or order :

Tocris Bioscience product webpage