Conantokin G | Tocris Bioscience 4136/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

Conantokin G

catalog :

4136/500

quantity :

500µg

price :

199 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

CCC(C)C(NC(=O)C(CC(C)C)NC(=O)C(CC(C(O)=O)C(O)=O)NC(=O)C(CCC(N)=O)NC(=O)C(CC(N)=O)NC(=O)C(CC(C(O)=O)C(O)=O)NC(=O)C(CCC(N)=O)NC(=O)C(CC(C)C)NC(=O)C(CC(C(O)=O)C(O)=O)NC(=O)C(CC(C(O)=O)C(O)=O)NC(=O)C(CCC(O)=O)NC(=O)CN)C(=O)NC(CCCNC(N)=N)C(=O)NC(CC(C(O)=O)C(O)=O)C(=O)NC(CCCCN)C(=O)NC(CO)C(=O)NC(CC(N)=O)C(N)=O

Cat Number :

4136/500

Product Name :

Conantokin G

Cas Number :

[93438-65-4]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

199 USD

Primary Category :

Ion Channels

Secondary Category :

Ligand-gated Ion Channels

Tertiary Category :

Glutamate (Ionotropic) Receptors

Primary Action :

NR2B-selective NMDA receptor antagonist

Biological Description :

NR2B-selective, competitive antagonist of the NMDA receptor. Blocks NMDA-evoked current in mouse cortical neurons (IC50 = 480 nM); also inhibits NMDA-evoked responses in oocytes expressing N2RB, but not NR2A, subunits (IC50 ~300 nM). Exhibits neuroprotective properties in vivo and in vitro.

Formula :

C88H138N26O44

Molwt :

2264.21

more info or order :

Tocris Bioscience product webpage