LY 266097 hydrochloride | Tocris Bioscience 4081/10 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

LY 266097 hydrochloride

catalog :

4081/10

quantity :

10 mg (also 50 mg)

price :

281 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
McCorvy J, Wacker D, Wang S, Agegnehu B, Liu J, Lansu K, et al. Structural determinants of 5-HT2B receptor activation and biased agonism. Nat Struct Mol Biol. 2018;25:787-796 pubmed publisher

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

4081

SKU :

4081/10

product name :

LY 266097 hydrochloride

Description :

Selective 5-HT2B antagonist

target :

5-HT2B Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

407.33

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

LY 266097 hydrochloride is a selective 5-HT2B receptor antagonist (pKi = 9.3). More than 100-fold selective over 5-HT2A and 5-HT2C. Attenuates amphetamine-induced locomotion in the rat.

extended description :

Selective 5-HT2B antagonist

chemical name text :

1-[(2-Chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,9-tetrahydro-6-methyl-1H-pyrido[3,4-b]indole hydrochloride

formula :

C 21 H 23 ClN 2 O 2 .HCl

formula text :

C21H23ClN2O2.HCl

cas num :

172895-39-5

USD :

281 USD

product details :

Selective 5-HT2B antagonist

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage