TCS 2510 | Tocris Bioscience 4069/1 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

TCS 2510

catalog :

4069/1

quantity :

1 mg

price :

285 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Zhang J, Vardy E, Muise E, Wang T, Visconti R, Vadlamudi A, et al. Utilizing Designed Receptors Exclusively Activated by Designer Drug Chemogenetic Tools to Identify Beneficial G Protein-Coupled Receptor Signaling for Fibrosis. J Pharmacol Exp Ther. 2020;375:357-366 pubmed publisher
Liu Y, Rajagopal M, Lee K, Battini L, Flores D, Gusella G, et al. Prostaglandin E(2) mediates proliferation and chloride secretion in ADPKD cystic renal epithelia. Am J Physiol Renal Physiol. 2012;303:F1425-34 pubmed publisher

product information

brand :

Tocris, a Bio-Techne Brand

catalog number base :

4069

SKU :

4069/1

product name :

TCS 2510

Description :

Selective EP4 agonist

target :

Prostanoid Receptor Agonists

category :

Small Molecules

unit size :

1 mg

purity :

98%

observed molecular weight :

383.49

url print :

?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM). Displays no significant binding at other prostaglandin receptors at concentrations up to 14 M.

extended description :

Selective EP4 agonist

chemical name text :

(5R)-5-[(3S)-3-Hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5-yl)hexyl]-2-pyrrolidinone

formula :

C 21 H 29 N 5 O 2

formula text :

C21H29N5O2

cas num :

346673-06-1

USD :

285 USD

product details :

Selective EP4 agonist

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage