MJ 15 | Tocris Bioscience 4063 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

MJ 15

catalog :

4063

quantity :

10 mg (also 50 mg)

price :

216 USD

more info or order :

Tocris Bioscience product webpage

citations: 2

Reference
Tan R, Cao L. Cannabinoid WIN-55,212-2 mesylate inhibits tumor necrosis factor-α-induced expression of nitric oxide synthase in dorsal root ganglion neurons. Int J Mol Med. 2018;42:919-925 pubmed publisher
Kong Y, Wang W, Zhang C, Wu Y, Liu Y, Zhou X. Cannabinoid WIN?55,212?2 mesylate inhibits ADAMTS?4 activity in human osteoarthritic articular chondrocytes by inhibiting expression of syndecan?1. Mol Med Rep. 2016;13:4569-76 pubmed publisher

product information

brand :

Tocris

master code :

4063

SKU :

4063/10

product name :

MJ 15

description :

Potent and selective CB1 antagonist

target :

Cannabinoid R1/CB1 Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

471.77

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Potent and selective CB1 receptor antagonist (Ki = 27.2 pM, IC50 = 118.9 pM for rat CB1 receptors). Exhibits potency in obesity and hyperlipidemia models; inhibits food intake and increases in body weight in diet-induced obese rats and mice.

catalog number base :

4063

product keywords :

MJ15 CB1 receptors antagonist cannabinoid receptors 1 antagonists obesity dyslipidemia dyslipidaemia CB1 Receptors 4063,

extended description :

Potent and selective CB1 antagonist

chemical name text :

5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(3-pyridinylmethyl)-1H-pyrazole-3-carboxamide

formula :

C 23 H 17 Cl 3 N 4 O

formula text :

C23H17Cl3N4O

cas num :

944154-76-1

2020 USD :

209

2021 USD :

216 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage