BMS 470539 dihydrochloride | Tocris Bioscience 4053/10 product information

This webpage contains legacy information. The product is either no longer available from the supplier or has been delisted at Labome.

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BMS 470539 dihydrochloride

catalog :

4053/10

quantity :

10 mg

price :

296 USD

citations: 1

Reference
Jain S, Panyutin A, Liu N, Xiao C, Pinol R, Pundir P, et al. Melanotan II causes hypothermia in mice by activation of mast cells and stimulation of histamine 1 receptors. Am J Physiol Endocrinol Metab. 2018;315:E357-E366 pubmed publisher

product information

brand :

Tocris

master code :

4053

SKU :

4053/10

product name :

BMS 470539 dihydrochloride

description :

Potent, selective MC1 receptor agonist

target :

Melanocortin Receptor Agonists

category :

Small Molecules

unit size :

10 mg

purity :

98%

observed molecular weight :

632.62

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

BMS 470539 dihydrochloride is a potent, selective melanocortin MC1 receptor agonist (IC50 = 120 nM). Exhibits anti-inflammatory properties following ischemia-reperfusion in the vasculature. Inhibits leukocyte trafficking.

catalog number base :

4053

extended description :

Potent, selective MC1 receptor agonist

chemical name text :

1-[1-(3-Methyl-L-histidyl-O-methyl-D-tyrosyl)-4-phenyl-4-piperidinyl]-1-butanone dihydrochloride

formula :

C 32 H 41 N 5 O 4 .2HCl

formula text :

C32H41N5O4.2HCl

cas num :

2341796-82-3

USD 2021 :

277

USD 2022 :

296 USD

product details :

Potent, selective MC1 receptor agonist

storage :

Desiccate at RT