Lisuride maleate | Tocris Bioscience 4052 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Lisuride maleate

catalog :

4052

quantity :

10 mg (also 50 mg)

price :

233 USD

more info or order :

Tocris Bioscience product webpage

citations: 3

Reference
Gadgaard C, Jensen A. Functional characterization of 5-HT1A and 5-HT1B serotonin receptor signaling through G-protein-activated inwardly rectifying K+ channels in a fluorescence-based membrane potential assay. Biochem Pharmacol. 2020;175:113870 pubmed publisher
McCorvy J, Wacker D, Wang S, Agegnehu B, Liu J, Lansu K, et al. Structural determinants of 5-HT2B receptor activation and biased agonism. Nat Struct Mol Biol. 2018;25:787-796 pubmed publisher
Chan J, Day T, Marchant J. Coalescing beneficial host and deleterious antiparasitic actions as an antischistosomal strategy. elife. 2018;7: pubmed publisher

product information

brand :

Tocris

master code :

4052

SKU :

4052/10

product name :

Lisuride maleate

description :

Dopamine agonist; antiparkinson's agent

target :

Non-selective Dopamine Receptor Agonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

454.52

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Dopamine receptor agonist and anti-Parkinson s agent. Displays high affinity for D2, D3 and D4 receptors along with 5-HT1A. Exhibits some 5-HT2B receptor antagonist properties. Decreases prolactin release; reduces inflammatory mediators such as TNF- and IL6. Exhibits anticonvulsive effects. Acts similar to bromocriptine (Cat. No. 0427).

catalog number base :

4052

product keywords :

antiparkinsonian drug anti-Parkinson s disease dopaminergic agonists dopamine receptor agonist DA Non-selective Dopamine Non-selective 5-HT 4052,

extended description :

Dopamine agonist; antiparkinson's agent

chemical name text :

N -[(8 )-9,10-Didehydro-6-methylergolin-8-yl]-N,N-diethylurea maleate

formula :

C 20 H 26 N 4 O.C 4 H 4 O 4

formula text :

C20H26N4O.C4H4O4

cas num :

19875-60-6

2020 USD :

224

2021 USD :

233 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage