CCG 63802 | Tocris Bioscience 4028 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

CCG 63802

catalog :

4028

quantity :

10 mg (also 50 mg)

price :

215 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Taccola G, Doyen P, Damblon J, Dingu N, Ballarin B, Steyaert A, et al. A new model of nerve injury in the rat reveals a role of Regulator of G protein Signaling 4 in tactile hypersensitivity. Exp Neurol. 2016;286:1-11 pubmed publisher

product information

brand :

Tocris

master code :

4028

SKU :

4028/10

product name :

CCG 63802

description :

Inhibitor of regulator of G-protein signaling 4 (RGS4) protein

target :

Regulators of G Protein Signaling (RGS) Inhibitors

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

450.51

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with G o. Retains activity under reducing conditions.

catalog number base :

4028

product keywords :

CCG63802 inhibitors inhibits regulator g-protein signaling signalling RGS RGS4 G proteins Heterotrimeric G-protein GTPases 4028,

extended description :

Inhibitor of regulator of G-protein signaling 4 (RGS4) protein

chemical name text :

(2E)-2-(1,3-Benzothiazol-2-yl)-3-[9-methyl-2-(3-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]acrylonitrile

formula :

C 26 H 18 N 4 O 2 S

formula text :

C26H18N4O2S

cas num :

620112-78-9

2020 USD :

210

2021 USD :

215 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage