ProTx II | Tocris Bioscience 4023/100 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

ProTx II

catalog :

4023/100

quantity :

100µg

price :

139 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

[H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@@H]3CSSC[C@H](NC(=O)[C@H](CC4=CNC5=C4C=CC=C5)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC4=CNC5=C4C=CC=C5)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC4=CNC5=C4C=CC=C5)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(N)=O)NC1=O)[C@@H](C)O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N3)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(O)=O)NC2=O)C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(O)=O

Cat Number :

4023/100

Product Name :

ProTx II

Cas Number :

[484598-36-9]

Unit Size :

100µg

Size :

100

Unit :

µg

USD :

139 USD

Primary Category :

Ion Channels

Secondary Category :

Sodium Channels

Tertiary Category :

Voltage-gated Sodium Channels

Primary Action :

Potent and selective NaV1.7 channel blocker

Biological Description :

Potent and selective NaV1.7 channel blocker (IC50 = 0.3 nM). Shifts activation gating positively and decreases current magnitude. Displays 100-fold selectivity over other sodium channel subtypes.

Formula :

C168H250N46O41S8

Molwt :

3826.59

more info or order :

Tocris Bioscience product webpage