JNJ 5207852 dihydrochloride | Tocris Bioscience 4020 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

JNJ 5207852 dihydrochloride

catalog :

4020

quantity :

10 mg (also 50 mg)

price :

195 USD

more info or order :

Tocris Bioscience product webpage

product information

brand :

Tocris

master code :

4020

SKU :

4020/10

product name :

JNJ 5207852 dihydrochloride

description :

High affinity H3 antagonist

target :

Histamine H3 Receptor Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

389.4

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity histamine H3 receptor neutral antagonist (pKi values are 8.9 and 9.2 in rat and human respectively). Brain penetrant and orally active. Has 3- and 100-fold higher affinity than thioperamide (Cat. No. 0644) for rat and human H3 receptors respectively. Suppresses slow-wave sleep; exhibits wake-promoting effects in rodent arousal models.

catalog number base :

4020

product keywords :

JNJ5207852 histamine receptor H3 neutral antagonist antagonists Histamine H3 Receptors 4020,

extended description :

High affinity H3 antagonist

chemical name text :

1-[3-[4-(1-Piperidinylmethyl)phenoxy]propyl]piperidine hydrochloride

formula :

C 20 H 32 N 2 O.2HCl

formula text :

C20H32N2O.2HCl

cas num :

1782228-76-5

2020 USD :

189

2021 USD :

195 USD

storage :

Desiccate at RT

more info or order :

Tocris Bioscience product webpage