MEN 11270 | Tocris Bioscience 3978/500 product information

product summary

request information :

company name :

Tocris Bioscience

product type :

chemical

product name :

MEN 11270

catalog :

3978/500

quantity :

500µg

price :

315 USD

more info or order :

Tocris Bioscience product webpage

product information

CHEMISTRY :

[H]N[C@H](CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC(=O)N[C@H](CC1=CC=CS1)C(=O)N[C@H]1CCNC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H]2CC3CCCCC3N2C(=O)[C@H]2CC3=CC=CC=C3CN2C1=O

Cat Number :

3978/500

Product Name :

MEN 11270

Cas Number :

[235082-52-7]

Unit Size :

500µg

Size :

500

Unit :

µg

USD :

315 USD

Primary Category :

7-TM Receptors

Secondary Category :

Peptide Receptors

Tertiary Category :

Bradykinin Receptors

Primary Action :

Selective B2 antagonist; analog of HOE 140 (Cat. No. 3014)

Biological Description :

Peptide antagonist of the B2 bradykinin receptor (pKi = 10.3); conformationally constrained cyclized analog of HOE 140 (Cat. No. 3014). Blocks hypotension and bronchoconstriction in vivo. Displays selectivity for B2 over 29 other receptors and ion channels (pIC50 < 5.5).

Formula :

C60H90N20O11S

Molwt :

1299.56

more info or order :

Tocris Bioscience product webpage