BCTC | Tocris Bioscience 3875 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BCTC

catalog :

3875

quantity :

10 mg (also 50 mg)

price :

169 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Lian Y, Cheng M, Zhang X, Wang L. Elevated expression of transient receptor potential vanilloid typeÂ 1 in dorsal root ganglia of rats with endometriosis. Mol Med Rep. 2017;16:1920-1926 pubmed publisher

product information

brand :

Tocris

master code :

3875

SKU :

3875/10

product name :

BCTC

description :

TRPV1 antagonist

target :

TRPV Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

372.89

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

Orally effective vanilloid receptor 1 (TRPV1 receptor) antagonist. Inhibits acid- and capsaicin-induced activation of rat TRPV1 receptors (IC50 values are 6.0 and 35 nM respectively). Displays analgesic properties in rat models of inflammatory and neuropathic pain. CNS penetrant.

catalog number base :

3875

product keywords :

vanilloid trpv1 antagonists transient receptors potential channels TRPV 3875,

extended description :

TRPV1 antagonist

chemical name text :

4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide

formula :

C 20 H 25 ClN 4 O

formula text :

C20H25ClN4O

cas num :

393514-24-4

2020 USD :

164

2021 USD :

169 USD

storage :

Store at RT

more info or order :

Tocris Bioscience product webpage