BL 1249 | Tocris Bioscience 3797 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

BL 1249

catalog :

3797

quantity :

10 mg (also 50 mg)

price :

190 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Fernández Fernández D, Cadaveira Mosquera A, Rueda Ruzafa L, Herrera Pérez S, Veale E, Reboreda A, et al. Activation of TREK currents by riluzole in three subgroups of cultured mouse nodose ganglion neurons. PLoS ONE. 2018;13:e0199282 pubmed publisher

product information

brand :

Tocris

master code :

3797

SKU :

3797/10

product name :

BL 1249

description :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) activator

target :

Two-P Potassium Channels Activators

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

99%

observed molecular weight :

291.35

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) channel opener (EC50 values are 5.5 M and 8 M, respectively). Exhibits selectivity for bladder over vascular tissue in vitro and in vivo (EC50 values are 1.26 and 21.0 M for cultured bladder and aortic tissues respectively).

catalog number base :

3797

product keywords :

BL1249 potassium channel activators openers K2p2.1 trek-1 kcnk2 tpkc1 bladder selective Two-P Potassium Channels 3797,

extended description :

K2P2.1 (TREK-1) and K2P10.1 (TREK-2) activator

chemical name text :

5,6,7,8-Tetrahydro-N-[2-(2H-tetrazol-5-yl)phenyl]-1-naphthalenamine

formula :

C 17 H 17 N 5

formula text :

C17H17N5

cas num :

18200-13-0

2020 USD :

182

2021 USD :

190 USD

storage :

Store at -20°C

more info or order :

Tocris Bioscience product webpage