Efonidipine hydrochloride monoethanolate | Tocris Bioscience 3733 product information

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product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

Efonidipine hydrochloride monoethanolate

catalog :

3733

quantity :

10 mg (also 50 mg)

price :

92 USD

product information

brand :

Tocris

SKU :

3733/10

product name :

Efonidipine hydrochloride monoethanolate

unit sizes :

10 mg (also 50 mg)

description :

CaV1.x and CaV3.x blocker

target :

Cav1.x Channel Blockers

category :

Small Molecules

purity :

99%

observed molecular weight :

714.18

details of functionality :

Selective blocker of L-type and T-type Ca2+ channels. Displays minimal inhibition of N- and P/Q-type channels and no inhibition of R-type channels. R (-) and S (+)-enantiomers display different channel selectivity; S (+)-Efonidipine blocks L-type and T-type channels whereas R (-)-Efonidipine displays selectivity for T-type channels. Exhibits antihypertensive activity.

catalog number base :

3733

extended description :

CaV1.x and CaV3.x blocker

chemical name text :

5-(5,5-Dimethyl-2-oxido-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3-pyridinecarboxylic acid 2-[phenyl(phenylmethyl)amino]ethyl ester hydrochloride monoethanolate

formula :

C 34 H 38 N 3 O 7 P.HCl.C 2 H 5 OH

formula text :

C34H38N3O7P.HCl.C2H5OH

cas num :

111011-76-8

USD :

92 USD

product details :

CaV1.x and CaV3.x blocker

storage :

Desiccate at +4°C