PF 514273 | Tocris Bioscience 3676 product information

product summary

company name :

Tocris Bioscience

product type :

chemical

product name :

PF 514273

catalog :

3676

quantity :

10 mg (also 50 mg)

price :

222 USD

more info or order :

Tocris Bioscience product webpage

citations: 1

Reference
Rozenfeld R, Gupta A, Gagnidze K, Lim M, Gomes I, Lee Ramos D, et al. AT1R-CB?R heteromerization reveals a new mechanism for the pathogenic properties of angiotensin II. EMBO J. 2011;30:2350-63 pubmed publisher

product information

brand :

Tocris

master code :

3676

SKU :

3676/10

product name :

PF 514273

description :

High affinity and selective CB1 antagonist

target :

Cannabinoid R1/CB1 Antagonists

category :

Small Molecules

unit size :

10 mg (also 50 mg)

purity :

98%

observed molecular weight :

452.28

url print :

?utm_source=distributor&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules

details of functionality :

High affinity and selective CB1 receptor antagonist (Ki values are 1 and 10000 nM at CB1 and CB2 receptors respectively). Inhibits food intake in vivo following oral administration.

catalog number base :

3676

product keywords :

Potent and selective CB1 agonists cannabinoids Receptors PF514273 cb1r CB1 Receptors 3676,

extended description :

High affinity and selective CB1 antagonist

chemical name text :

2-(2-Chlorophenyl)-3-(4-chlorophenyl)-7-(2,2-difluoropropyl)-6,7-dihydro-2H-pyrazolo[3,4-f][1,4]oxazepin-8(5H)-one

formula :

C 21 H 17 Cl 2 F 2 N 3 O 2

formula text :

C21H17Cl2F2N3O2

cas num :

851728-60-4

2020 USD :

215

2021 USD :

222 USD

storage :

Store at +4°C

more info or order :

Tocris Bioscience product webpage